PROCESS FOR PREPARING 2-CHLOROTHIAZOLE COMPOLUNDS
Application 2499/DEL/2004 published 2006-11-17, filed 2004-12-15
The invention relates to a process for preparing a compound of formula (I), in which X is CH or N, Y is NO2 or CN, Z is CHR3, O, NR3 or S, R1 and R2 are either each, independently of the other, hydrogen or unsubstituted or R4substituted alkyl or together a two- or three-membered alkylene bridge or a two- or three-membered alkylene bridge in which one member is replaced by a hetero member selected from the group, consisting of NR5, O and S, R3 is H or unsubstituted or R4-substituted alkyl, R4 is an unsubstituted or substituted aryl or heteroaryl group, and R5 is H or alkyl, which comprises a) reacting a compound of formula (II) with a chlorinating agent or b1) initially reacting a compound of formula (IV) with a compound of formula (V) and b2) further reacting the compound of formula (II) obtainable thereby, with or without intermediate isolation, with a chlorinating agent, to intermediates used in this process, to the use of these intermediates and to a process for the preparation of these intermediates.
Applicant
1)SYNGENTA PARTICIPATIONS AG
:SCHWARZWALDALLEE 215, CH-4058 BASEL, SWITZERLAND Switzerland
Inventor
1)HENRY SZCZEPANSKI 2)THOMAS GOBEL 3)OTTMAN FRANZ HUTER 4)ANTHONY CORNELIUS O'SULLIVAN 5)MARCEL SENN 6)THOMAS RAPOLD 7)PETER MAIENFISCH 8)THOMAS PITTERNA
International Info
Classification: C07D277/32
Priority Information
3412/95 Switzerland 1995-12-01