TACHYKININ RECEPTOR ANTAGONISTS
Application 1604/KOLNP/2004 published 2006-08-11, filed 2004-10-26
The present invention relates to selective NK-1 receptor antagonists of Formula (I); or a pharmaceutically acceptable salt thereof, for the treatment of disorders associated with an excess of tachykinins. (FIG. 1)
Applicant
ELI LILLY AND COMPANY
LILLY CORPORATE CENTER, INDIANAPOLIS, IN 46285, UNITED STATES OF AMERICA
Inventor
AMEGADZIE, ALBERT KUDZOVI; GARDINIER, KEVIN, MATTHEW; HEMBRE, ERIK, JAMES; HONG, JIAN, ERIC; JUNGHEIM, LOUIS, NICKOLAUS; MUEHL, BRIAN, STEPHEN; REMICK, DAVID, MICHAEL; ROBERTSON, MICHAEL, ALAN; SAVIN, KENNETH, ALLEN
International Info
Classification: C07D 249/06
Publication Number: WO 03/091227
Application Date: 2003-04-22
Priority Information
60/376,121 USA 2002-04-26
60/440,865 USA 2002-01-16