VITAMIN D RECEPTOR MODULATORS
Application 1191/KOLNP/2005 published 2006-07-21, filed 2005-06-21
The present invention relates to novel, non-secosteroidal, diaryl compounds with vitamin D receptor (VDR) modulating activity that are less hypercalcemic than 1a,25 dihydroxy vitamin D3. These compounds are useful for treating bone disease and psoriasis (FIG. - nil)
Applicant
ELI LILLY AND COMPANY
LILLY CORPORATE CENTER INDIANAPOLIS IN 46285 USA
Inventor
1. EMILIO ENRIQUE BUNEL 2. ROBERT PETER GAJEWSKI 3. CHARLES DAVID JONES 4. JIANLIANG LU 5. TIQNWEI MA 6. SUNIL NAGPAL 7. YING KWONG YEE
International Info
Classification: C07C 59/90,62/24,69/78,235/34,311/50,317/28,C07D 257/06,277/34,A61K 31/12,31/65,31/18,31/19,31/192,31/235,31/41,31/426
Publication Number: WO 04/048309 A1
Application Date: 2003-11-20
Priority Information
60/429,041 US 2003-11-22