PHENYL-THIOPHENE TYPE VITAMIN D RECEPTOR MODULATORS
Application 1967/KOLNP/2004 published 2006-11-03, filed 2004-12-21
The present invention relates to novel, non-secosteroidal, phenyl-thiophene compounds with vitamin D receptor (VDR) modulating DFWLYLW\WKDWDUHOHVVK\SHUFDOFHPLFWKDQ.GLK\GUR[\YLWDPLQ'7KHVHFRPSRXQGVDUHXVHIXOIRUWUHDWLQJERQHGLVHDVHDQGpsoriasis. (FIG.nil)
Applicant
ELI LILLY AND COMPANY.,
LILLY CORPORATE CENTER, INDIANAPOLIS, IN 46285, USA.
Inventor
DAHNKE, KARL, ROBERT GAJEWSKI, ROBERT, PETER JONES, CHARLES, DAVID LINEBARGER, JARED, HARRIS LU, JIANLIANG MA, TIANWEI NAGPAL, SUNIL SIMARD, TODD, PARKER TEE, TING, KWONG BUNEL, EMILIO, ENRIQUE STITES, RYAN, EDWARD
International Info
Classification: C07D 333/38, 333/16, 333/18, 333/22, 409/12, 409/06, 333/34, 413/04, 409/04, A61K 31/381, 31/401, 31/41, 31/4245, A61P
Publication Number: WO 03/101978
Application Date: 2003-05-22
Priority Information
60/384,151 USA 2002-05-29